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SB 742457

CAS No. 607742-69-8

SB 742457 ( GSK742457 )

产品货号. M15279 CAS No. 607742-69-8

SB742457 is a highly selective 5-HT6 receptor antagonist with pKi of 9.63.

纯度: >98%(HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
5MG ¥551 有现货
10MG ¥883 有现货
25MG ¥1798 有现货
50MG ¥2876 有现货
100MG ¥4560 有现货
500MG ¥9558 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    SB 742457
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    SB742457 is a highly selective 5-HT6 receptor antagonist with pKi of 9.63.
  • 产品描述
    SB742457 is a highly selective 5-HT6 receptor antagonist with pKi of 9.63, exhibits >100-fold selectivity over other receptors. Phase 2.
  • 同义词
    GSK742457
  • 通路
    Endocrinology/Hormones
  • 靶点
    5-HT Receptor
  • 受体
    5-HT6
  • 研究领域
    Neurological Disease
  • 适应症
    ——

化学信息

  • CAS Number
    607742-69-8
  • 分子量
    353.44
  • 分子式
    C19H19N3O2S
  • 纯度
    >98%(HPLC)
  • 溶解度
    Ethanol: 2 mg/mL (5.65 mM); DMSO: 78 mg/mL (220.68 mM)
  • SMILES
    O=S(C1=CC2=CC=CC(N3CCNCC3)=C2N=C1)(C4=CC=CC=C4)=O
  • 化学全称
    3-Phenylsulfonyl-8-(piperazin-1-yl)quinoline

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1.Chuang ATT, et al. Alzheimers Dement, 2006, 2, S631–S632 (abstract).
产品手册
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