SB 742457
CAS No. 607742-69-8
SB 742457 ( GSK742457 )
产品货号. M15279 CAS No. 607742-69-8
SB742457 is a highly selective 5-HT6 receptor antagonist with pKi of 9.63.
纯度: >98%(HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥551 | 有现货 |
|
10MG | ¥883 | 有现货 |
|
25MG | ¥1798 | 有现货 |
|
50MG | ¥2876 | 有现货 |
|
100MG | ¥4560 | 有现货 |
|
500MG | ¥9558 | 有现货 |
|
1G | 获取报价 | 有现货 |
|
生物学信息
-
产品名称SB 742457
-
注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
-
产品简述SB742457 is a highly selective 5-HT6 receptor antagonist with pKi of 9.63.
-
产品描述SB742457 is a highly selective 5-HT6 receptor antagonist with pKi of 9.63, exhibits >100-fold selectivity over other receptors. Phase 2.
-
同义词GSK742457
-
通路Endocrinology/Hormones
-
靶点5-HT Receptor
-
受体5-HT6
-
研究领域Neurological Disease
-
适应症——
化学信息
-
CAS Number607742-69-8
-
分子量353.44
-
分子式C19H19N3O2S
-
纯度>98%(HPLC)
-
溶解度Ethanol: 2 mg/mL (5.65 mM); DMSO: 78 mg/mL (220.68 mM)
-
SMILESO=S(C1=CC2=CC=CC(N3CCNCC3)=C2N=C1)(C4=CC=CC=C4)=O
-
化学全称3-Phenylsulfonyl-8-(piperazin-1-yl)quinoline
运输与储存
-
储存条件(-20℃)
-
运输条件With Ice Pack
-
稳定性≥ 2 years
参考文献
1.Chuang ATT, et al. Alzheimers Dement, 2006, 2, S631–S632 (abstract).
产品手册
关联产品
-
Amitriptyline hydroc...
Amitriptyline Hydrochloride is a dibenzocycloheptene-derivative tricyclic antidepressant (TCA).
-
Pimavanserin
Pimavanserin(ACP-103) is a potent and selective 5-HT2A receptor inverse agonist with mean pIC50 of with 8.7 in the cell-based functional assay.
-
Escitalopram
Escitalopram is a selective serotonin reuptake inhibitor (SSRI) with Ki of 0.89 nM.